Raphael Volpert

Quantifying the effect of nootropics on cognitive performance using brain organoids.

Objective

  • Measure the effect of experimental nootropics such as PRL-8-53, Idra-21 and Lion's Mane on human cognitive performance using brain organoids.

  • Creating the first standardized neurochemical benchmark for cognitive enhancers “Nootropic-Analysis“.

  • Discover the optimal blueprint of compounds to decrease tolerance buildup and volatility from baseline while still enhancing cognition.

Motivation

  • Progress in discovering compounds which enhance brain health and performance has been held back by two bottlenecks:

    • Limited functional neuroimaging, both metabolic and electrical, and fMRI, is not a good marker for the neurochemical effects of compounds.

    • The slow turnaround of rodent and primate studies.

  • Building an automated brain organoid facility removes both barriers:

    • Because the tissue is exposed rather than encased, we can directly couple it to microscopes, multi-electrode arrays, optical reporters, and metabolic assays.

    • Scale of labautomation: allowing to run hundreds of “drug discovery-runs” instead of needing to do manual liquid handling, optical readout and data analysis for just a single one.

Milestones

  • In the first 3 months of Calculus, I am developing an open-source and highly modular version of the Cortical Labs CL1, focusing on the two hardest parts: the perfusion system and microelectrode array.

  • After setting up the infrastructure, I will start my first “Benchmarking-Run“ on the Lion's Mane compound and measure the ability of the organoids to solve problems.

  • Record baseline electrophysiology with multi-electrode arrays, track calcium dynamics, and capture transcriptomic profiles.

  • Monitor changes in synaptic-plasticity markers (BDNF, phosphorylated CREB), histone acetylation levels, and network oscillations linked to memory.

Raphael Volpert

Quantifying the effect of nootropics on cognitive performance using brain organoids.

Objective

  • Measure the effect of experimental nootropics such as PRL-8-53, Idra-21 and Lion's Mane on human cognitive performance using brain organoids.

  • Creating the first standardized neurochemical benchmark for cognitive enhancers “Nootropic-Analysis“.

  • Discover the optimal blueprint of compounds to decrease tolerance buildup and volatility from baseline while still enhancing cognition.

Motivation

  • Progress in discovering compounds which enhance brain health and performance has been held back by two bottlenecks:

    • Limited functional neuroimaging, both metabolic and electrical, and fMRI, is not a good marker for the neurochemical effects of compounds.

    • The slow turnaround of rodent and primate studies.

  • Building an automated brain organoid facility removes both barriers:

    • Because the tissue is exposed rather than encased, we can directly couple it to microscopes, multi-electrode arrays, optical reporters, and metabolic assays.

    • Scale of labautomation: allowing to run hundreds of “drug discovery-runs” instead of needing to do manual liquid handling, optical readout and data analysis for just a single one.

Milestones

  • In the first 3 months of Calculus, I am developing an open-source and highly modular version of the Cortical Labs CL1, focusing on the two hardest parts: the perfusion system and microelectrode array.

  • After setting up the infrastructure, I will start my first “Benchmarking-Run“ on the Lion's Mane compound and measure the ability of the organoids to solve problems.

  • Record baseline electrophysiology with multi-electrode arrays, track calcium dynamics, and capture transcriptomic profiles.

  • Monitor changes in synaptic-plasticity markers (BDNF, phosphorylated CREB), histone acetylation levels, and network oscillations linked to memory.

Raphael Volpert

Quantifying the effect of nootropics on cognitive performance using brain organoids.

Objective

  • Measure the effect of experimental nootropics such as PRL-8-53, Idra-21 and Lion's Mane on human cognitive performance using brain organoids.

  • Creating the first standardized neurochemical benchmark for cognitive enhancers “Nootropic-Analysis“.

  • Discover the optimal blueprint of compounds to decrease tolerance buildup and volatility from baseline while still enhancing cognition.

Motivation

  • Progress in discovering compounds which enhance brain health and performance has been held back by two bottlenecks:

    • Limited functional neuroimaging, both metabolic and electrical, and fMRI, is not a good marker for the neurochemical effects of compounds.

    • The slow turnaround of rodent and primate studies.

  • Building an automated brain organoid facility removes both barriers:

    • Because the tissue is exposed rather than encased, we can directly couple it to microscopes, multi-electrode arrays, optical reporters, and metabolic assays.

    • Scale of labautomation: allowing to run hundreds of “drug discovery-runs” instead of needing to do manual liquid handling, optical readout and data analysis for just a single one.

Milestones

  • In the first 3 months of Calculus, I am developing an open-source and highly modular version of the Cortical Labs CL1, focusing on the two hardest parts: the perfusion system and microelectrode array.

  • After setting up the infrastructure, I will start my first “Benchmarking-Run“ on the Lion's Mane compound and measure the ability of the organoids to solve problems.

  • Record baseline electrophysiology with multi-electrode arrays, track calcium dynamics, and capture transcriptomic profiles.

  • Monitor changes in synaptic-plasticity markers (BDNF, phosphorylated CREB), histone acetylation levels, and network oscillations linked to memory.